WebMay 1, 2007 · Substituted oxathiolone fused chalcones were prepared by condensation of 4-acetyl-5-methoxy-2-oxo-benz[1,3]oxathiole with benzaldehydes under acidic … WebAug 5, 2015 · Three structurally related oxathiolone fused chalcone derivatives appeared effective chemosensitizers, able to restore in part sensitivity to fluconazole of multidrug-resistant C. albicans strains. Compound 21 effectively chemosensitized cells resistant due to the overexpression of the MDR1 gene, compound 6 reduced resistance of cells …
1,2-Oxathiolane, 2,2-dioxide - NIST
WebJun 1, 2007 · Oxathiolone-fused chalcones Antibacterial [11]Neohesperidin dihydrochalcone Antioxidant [12] Chalcone-based bisulfones and sulfones Antifungal [13] Naphthalenyl and pyridinyl analogs... WebSep 1, 2011 · Summary AMG‐148, an oxathiolone‐fused chalcone derivative, exhibited in vitro antifungal activity against several strains of human pathogenic yeast, with minimum inhibitory concentration values within the range of 1–16 μg ml−1 and a fungicidal effect was observed at higher concentrations. Presence of major drug‐effluxing membrane proteins … thursday night football game today
Synthesis of Isomeric, Oxathiolone Fused Chalcones, and …
WebSubstituted oxathiolone fused chalcones were prepared by condensation of 4-acetyl-5-methoxy-2-oxo-benz[1,3]oxathiole with benzaldehydes under acidic conditions. The compounds were tested for cytotoxic, antibacterial, antifungal and tuberculostatic activity. Three derivatives demonstrated weak activity against HeLa cells, two were slightly active … WebAbstract AMG-148, an oxathiolone-fused chalcone derivative, exhibited in vitro antifungal activity against several strains of human pathogenic yeast, with minimum inhibitory concentration values within the range of 1-16 μg ml (-1) and a fungicidal effect was observed at higher concentrations. WebAug 5, 2015 · Three structurally related oxathiolone fused chalcone derivatives appeared effective chemosensitizers, able to restore in part sensitivity to fluconazole of multidrug … thursday night football game week 18